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050 0 0 _aRS420
_b.T49 20117
245 0 0 _aTextbook of drug design and discovery /
_cedited by Povl Krogsgaard-Larsen, Kristian Strømgaard, Ulf Madsen.
250 _a5th ed.
260 _aBoca Raton, FL :
_bCRC Press/Taylor & Francis,
_c2017
300 _axiii 436 p.
504 _aIncludes bibliographical references and index.
505 0 _aMolecular recognition in ligand-protein binding / Tommy Liljefors -- Biostructure-based drug design / Flemming S. Jørgensen and Jette S. Kastrup -- Ligand-based drug design / Ingrid Pettersson, Thomas Balle, and Tommy Liljefors -- Chemical biology / Kristian Strømgaard -- Stereochemistry in drug design / M. Belen Mayo-Martin and David E. Jane -- Natural products in drug discovery / Guy T. Carter -- Imaging in drug discovery and development / Markus Rudin and Thomas Mueggler -- Peptides and peptidomimetics / Minying Cai, Vinod Kulkarni, and Victor J. Hruby -- Prodrugs : design and development / Anders Buur and Niels Mørk -- Metals in medicine : inorganic medicinal chemistry / Helle R. Hansen and Ole Farver -- Enzyme inhibitors : biostructure-based and mechanism-based designs / Robert A. Copeland, Richard R. Gontarek, and Lusong Luo -- Receptors : structure, function, and pharmacology / Hans Bräuner-Osborne -- Ion channels : structure and function / Søren-Peter Olesen and Daniel B. Timmermann -- Neurotransmitter transporters : structure and function / Claus J. Loland and Ulrik Gether -- GABA and glutamic acid receptor ligands / Bente Frølund and Ulf Madsen -- Acetylcholine / Anders A. Jensen and Povl Krogsgaard-Larsen -- Histamine receptors / Iwan de Esch, Henk Timmerman and Rob Leurs -- Dopamine and serotonin / Benny Bang-Andersen and Klaus P. Bøgesø -- Opioid and cannabinoid receptors / Rasmus P. Clausen and Harald S. Hansen -- Hypnotics / Bjarke Ebert and Keith Wafford -- Neglected diseases / Søren B. Christensen -- Immunomodulating agents / Ulla G. Sidelmann -- Anticancer agents / Fredrik Bjørkling and Lars H. Jensen -- Antiviral drugs / Erik De Clercq -- Antibiotics / Piet Herdewijn.
650 0 _aDrugs
_xDesign.
650 1 2 _aDrug Design.
650 2 2 _aDrug Discovery.
700 1 _aKrogsgaard-Larsen, Povl.
700 1 _aStrømgaard, Kristian.
700 1 _aMadsen, Ulf.
906 _a7
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999 _c20012
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